Cu-catalyzed cross-dehydrogenative coupling of the C7 C-H bond of indolines with sulfoximines has been accomplished. The reaction can be extended to the cross-dehydrogenative coupling of N-aryl 7-azaindoles with monoselectivity. The… Click to show full abstract
Cu-catalyzed cross-dehydrogenative coupling of the C7 C-H bond of indolines with sulfoximines has been accomplished. The reaction can be extended to the cross-dehydrogenative coupling of N-aryl 7-azaindoles with monoselectivity. The use of first-row copper catalysis, substrate scope, and late-stage synthetic applications are the important practical features.
Keywords:
dehydrogenative coupling;
copper catalyzed;
indolines sulfoximines;
cross dehydrogenative
Journal Title: Organic letters
Year Published: 2022
Link to full text (if available)
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Journal Title: Organic letters
Year Published: 2022
Link to full text (if available)
Share on Social Media: Sign Up to like & get
recommendations!