A mild and efficient method for the copper-catalyzed diamination of alkenes is described. In this reaction, o-benzoylhydroxylamine serves as an electrophilic nitrogen source for the regioselective formation of C-N bonds.… Click to show full abstract
A mild and efficient method for the copper-catalyzed diamination of alkenes is described. In this reaction, o-benzoylhydroxylamine serves as an electrophilic nitrogen source for the regioselective formation of C-N bonds. This transformation provides a novel strategy for synthesizing all four isomeric 2,3-disubstituted azaindoline families and offers a wide substrate scope.
Keywords:
alkenes using;
azaindoline families;
diamination alkenes;
catalyzed diamination;
copper catalyzed
Journal Title: Organic letters
Year Published: 2024
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Journal Title: Organic letters
Year Published: 2024
Link to full text (if available)
Share on Social Media: Sign Up to like & get
recommendations!