An efficient protocol to construct spiro[indole-3,4'-pyrazol]-5'-ones via ruthenium(II)-catalyzed selective C-H bond activation/[4 + 1] spirocyclization starting from easily available N-aryl amidines and diazopyrazolones has been developed. A series of spiro-pyrazolones... Click to show full abstract
An efficient protocol to construct spiro[indole-3,4'-pyrazol]-5'-ones via ruthenium(II)-catalyzed selective C-H bond activation/[4 + 1] spirocyclization starting from easily available N-aryl amidines and diazopyrazolones has been developed. A series of spiro-pyrazolones...
               
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