Articles with "acetamide linker" as a keyword



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Novel benzenesulfonamide‐thiouracil conjugates with a flexible N‐ethyl acetamide linker as selective CA IX and CA XII inhibitors

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Published in 2022 at "Archiv der Pharmazie"

DOI: 10.1002/ardp.202200434

Abstract: Novel benzenesulfonamide derivatives linked to diverse functionalized thiouracils through a flexible N‐ethyl acetamide linker were designed and synthesized as carbonic anhydrase (CA) inhibitors. The synthesized candidates demonstrated a potent inhibitory activity against four different CA… read more here.

Keywords: novel benzenesulfonamide; xii; acetamide linker; linker ... See more keywords