Synthesis and antimicrobial evaluation of piperic acid amides and their lower homologues
Sign Up to like & getrecommendations! Published in 2019 at "Drug Development Research"
DOI: 10.1002/ddr.21630
Abstract: Seven piperic acid amides along with their lower homologs (12) were synthesized using HATU‐DIPEA coupling reagent. All the synthesized derivatives were evaluated for their antibacterial activities against Staphylococcus aureus, Pseudomonas aeruginosa, and vancomycin‐resistant P. aeruginosa.… read more here.
Keywords: acid amides; piperic acid; found active; synthesis antimicrobial ... See more keywords
Fatty acid amides as potential circulating biomarkers for sarcopenia
Sign Up to like & getrecommendations! Published in 2023 at "Journal of Cachexia, Sarcopenia and Muscle"
DOI: 10.1002/jcsm.13244
Abstract: Sarcopenia is characterized by a progressive decrease in skeletal muscle mass and function with age. Given that sarcopenia is associated with various metabolic disorders, effective metabolic biomarkers for its early detection are required. We aimed… read more here.
Keywords: amides potential; potential circulating; acid amides; circulating biomarkers ... See more keywords
Ultrasound-assisted green bromination of N-cinnamoyl amino acid amides – Structural characterization and antimicrobial evaluation
Sign Up to like & getrecommendations! Published in 2017 at "Journal of Molecular Structure"
DOI: 10.1016/j.molstruc.2017.01.056
Abstract: Abstract N -phenylpropenoyl amino acid amides have been brominated using two alternative sonochemically activated green chemistry procedures. The first synthetic procedure has involved an ultrasound assisted bromination in an aqueous medium using ionic liquid as… read more here.
Keywords: ultrasound assisted; bromination; amino acid; acid amides ... See more keywords
Toporosides A and B, Cyclopentenyl-Containing ω-Glycosylated Fatty Acid Amides, and Toporosides C and D from the Northwestern Pacific Marine Sponge Stelodoryx toporoki.
Sign Up to like & getrecommendations! Published in 2022 at "Journal of natural products"
DOI: 10.1021/acs.jnatprod.2c00130
Abstract: Toporosides A-D (1-4), new ω-glycosylated fatty acid amides, were isolated from the sponge Stelodoryx toporoki. The structures of these compounds, including absolute configurations of stereogenic centers, were established using analysis of 1D and 2D NMR,… read more here.
Keywords: sponge stelodoryx; stelodoryx toporoki; acid amides; glycosylated fatty ... See more keywords
Multicomponent Approach to Libraries of Substituted Dihydroorotic Acid Amides.
Sign Up to like & getrecommendations! Published in 2019 at "ACS combinatorial science"
DOI: 10.1021/acscombsci.9b00144
Abstract: A process featuring a sequential multicomponent reaction followed by regioselective post-cyclization strategy was implemented for the facile synthesis of N,N'-disubstituted dihydroorotic acid amides in very mild condition. We obtained, for the first time, a library… read more here.
Keywords: approach libraries; acid amides; multicomponent approach; dihydroorotic acid ... See more keywords
Phosphorylation of Oxyethylated Calix[4]resorcinols with Phosphorous Acid Amides
Sign Up to like & getrecommendations! Published in 2018 at "Russian Journal of General Chemistry"
DOI: 10.1134/s1070363218010255
Abstract: The reaction of octa-2-hydroxyethylated calix[4]resorcinols with phosphorous acid amides and the subsequent thionylation by elemental sulfur afforded hydrolytically stable oxyethyl calix[4]resorcinols containing eight thiophosphoryl fragments. read more here.
Keywords: acid amides; resorcinols phosphorous; calix resorcinols; phosphorous acid ... See more keywords
Qualitative and Quantitative Analysis of Six Fatty Acid Amides in 11 Edible Vegetable Oils Using Liquid Chromatography–Mass Spectrometry
Sign Up to like & getrecommendations! Published in 2022 at "Frontiers in Nutrition"
DOI: 10.3389/fnut.2022.857858
Abstract: Fatty acid amides (FAAs) are endogenous lipid molecules that exhibit various physiological activities. FAAs are usually present at nanomolar levels in biological samples. In this study, a method for the qualitative and quantitative determination of… read more here.
Keywords: oil; qualitative quantitative; vegetable oils; edible vegetable ... See more keywords
Lithocholic Acid Amides as Potent Vitamin D Receptor Agonists
Sign Up to like & getrecommendations! Published in 2022 at "Biomolecules"
DOI: 10.3390/biom12010130
Abstract: 1α,25-Dihydroxyvitamin D3 [1α,25(OH)2D3, 1] is an active form of vitamin D3 and regulates various biological phenomena, including calcium and phosphate homeostasis, bone metabolism, and immune response via binding to and activation of vitamin D receptor… read more here.
Keywords: lithocholic acid; vitamin receptor; amides potent; acid amides ... See more keywords
Enzymatic Synthesis of 2-Chloropurine Arabinonucleosides with Chiral Amino Acid Amides at the C6 Position and an Evaluation of Antiproliferative Activity In Vitro
Sign Up to like & getrecommendations! Published in 2023 at "International Journal of Molecular Sciences"
DOI: 10.3390/ijms24076223
Abstract: A number of purine arabinosides containing chiral amino acid amides at the C6 position of the purine were synthesized using a transglycosylation reaction with recombinant E. coli nucleoside phosphorylases. Arsenolysis of 2-chloropurine ribosides with chiral… read more here.
Keywords: chiral amino; amino acid; synthesis; acid amides ... See more keywords
Synthesis, Quantification, and Characterization of Fatty Acid Amides from In Vitro and In Vivo Sources
Sign Up to like & getrecommendations! Published in 2021 at "Molecules"
DOI: 10.3390/molecules26092543
Abstract: Fatty acid amides are a diverse family of underappreciated, biologically occurring lipids. Herein, the methods for the chemical synthesis and subsequent characterization of specific members of the fatty acid amide family are described. The synthetically… read more here.
Keywords: acid amides; fatty acid; quantification; characterization ... See more keywords