Residency time of agonists does not affect the stability of GPCR–arrestin complexes
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DOI: 10.1111/bph.15846
Abstract: The interaction of arrestins with G‐protein coupled receptors (GPCRs) desensitizes agonist‐dependent receptor responses and often leads to receptor internalization. GPCRs that internalize without arrestin have been classified as “class A” GPCRs whereas “class B” GPCRs… read more here.
Keywords: agonists affect; residency time; affect stability; arrestin ... See more keywords