Loop‐F of the &agr;‐subunit determines the pharmacologic profile of novel competitive inhibitors of GABAA receptors
Sign Up to like & getrecommendations! Published in 2017 at "European Journal of Pharmacology"
DOI: 10.1016/j.ejphar.2017.01.033
Abstract: ABSTRACT The neurotransmitter &ggr;‐amino butyric acid (GABA) has a fundamental role in CNS function and ionotropic (GABAA) receptors that mediate many of the actions of GABA are important therapeutic targets. This study reports the mechanism… read more here.
Keywords: gabaa receptors; agr subunit; loop agr;