Iridium-Catalyzed Regio- and Enantioselective N-Allylation of Pyrazoles with Dienyl/Monoallylic Alcohols.
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DOI: 10.1021/acs.orglett.4c01201
Abstract: Here we report the first example of iridium-catalyzed asymmetric N-allylation of pyrazoles with dienyl allylic alcohols under mild conditions with broad functional group tolerance, exhibiting excellent N1/C3-site selectivities and enantioselectivities (up to >99% ee). In… read more here.
Keywords: catalyzed regio; iridium catalyzed; allylation pyrazoles; regio enantioselective ... See more keywords