Discovery of new 6-ureido/amidocoumarins as highly potent and selective inhibitors for the tumour-relevant carbonic anhydrases IX and XII
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DOI: 10.1080/14756366.2022.2154603
Abstract: Abstract A series of 6-ureido/amidocoumarins (5a–p and 7a–c) has been designed and synthesised to develop potent and isoform- selective carbonic anhydrase hCA XI and XII inhibitors. All coumarin derivatives were investigated for their CA inhibitory… read more here.
Keywords: ureido amidocoumarins; discovery new; new ureido; hca xii ... See more keywords