In vitro Antibacterial Evaluation of 1,2,4-Triazole Compounds Containing Purine Moiety
Sign Up to like & getrecommendations! Published in 2017 at "Chemistry of Natural Compounds"
DOI: 10.1007/s10600-017-2217-7
Abstract: 9H-[1,2,4]Triazolo[4,3-g]purin-5-amine (2) was synthesized by reaction of 6-hydrazinyl-7H-purin-2-amine (1a) with formic acid under reflux conditions. Treating compound 1a in ethanol with CS2 in the presence of KOH yielded 5-amino-3H-[1,2,4]triazolo[4,3-g]purine-3-thione (3). The new synthesized compounds were… read more here.
Keywords: containing purine; evaluation triazole; triazole compounds; compounds containing ... See more keywords
Synthesis and antibacterial evaluation of diaminomaleonitrile-based azo-Schiff bases and 8,9-dihydro-7H-purine-6-carboxamides
Sign Up to like & getrecommendations! Published in 2020 at "Research on Chemical Intermediates"
DOI: 10.1007/s11164-020-04175-y
Abstract: Some new DAMN-based Schiff base 6a–6g were synthesized via a condensation reaction of the corresponding azo dyes with 1-(2-amino-1,2-dicyanovinyl)-3-phenylurea. In continuation, facile synthesis of new 8,9-dihydro-7H-purine-6-carboxamide 7a–7g was reported via an efficient reaction of azo… read more here.
Keywords: synthesis antibacterial; dihydro purine; based azo; diaminomaleonitrile based ... See more keywords
Synthesis and antibacterial evaluation of (E)-1-(1H-indol-3-yl) ethanone O-benzyl oxime derivatives against MRSA and VRSA strains.
Sign Up to like & getrecommendations! Published in 2021 at "Bioorganic chemistry"
DOI: 10.1016/j.bioorg.2021.105288
Abstract: Infections caused due to multidrug resistant organisms have emerged as a constant menace to human health. Even though numerous antibiotics are currently available for treating infectious diseases, a great number of bacterial strains have acquired… read more here.
Keywords: evaluation indol; indol ethanone; synthesis antibacterial; mrsa vrsa ... See more keywords
Design, Synthesis, Antibacterial Evaluation, Three-Dimensional Quantitative Structure-Activity Relationship, and Mechanism of Novel Quinazolinone Derivatives.
Sign Up to like & getrecommendations! Published in 2023 at "Journal of agricultural and food chemistry"
DOI: 10.1021/acs.jafc.2c07264
Abstract: Plant bacterial illnesses are common and cause dramatic damage to agricultural goods all over the world, yet there are few efficient bactericides to alleviate them at present. To discover novel antibacterial agents, two series of… read more here.
Keywords: design synthesis; mechanism; quinazolinone derivatives; antibacterial evaluation ... See more keywords
Synthesis and Antibacterial Evaluation of Benzofuran Based Di-1,2,3-triazoles
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DOI: 10.1134/s1070363218070265
Abstract: A series of novel benzofuran-1,2,3-triazole hybrid molecules are synthesized using the click chemistry approach. Structures of the synthesized compounds were assessed by IR, NMR, and mass spectroscopy. The tests of final products 10a–10l for their… read more here.
Keywords: synthesis antibacterial; evaluation benzofuran; based triazoles; chemistry ... See more keywords
Antibacterial Evaluation, In Silico Characters and Molecular Docking of Schiff Bases Derived from 5-aminopyrazoles
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DOI: 10.3390/molecules24173130
Abstract: A series of Schiff bases 14–25 were designed and synthesized for evaluation of their antibacterial properties against multi-drug resistant bacteria (MDRB). The antibacterial activities of Schiff bases 14–25 showed that most of the synthesized compounds… read more here.
Keywords: schiff; schiff bases; silico; antibacterial evaluation ... See more keywords
Extraction and antibacterial evaluation of marine AMPs against diabetic wound pathogens
Sign Up to like & getrecommendations! Published in 2020 at "journal of applied pharmaceutical science"
DOI: 10.7324/japs.2020.101112
Abstract: The need for an alternative wound dressing material with effective coatings using antimicrobial peptides (AMPs) from a marine fish (Carangoides malabaricus) was selected as the primary objective in the present research. The AMPs were extracted… read more here.
Keywords: dressing material; wound dressing; evaluation marine; marine amps ... See more keywords