Beyond cysteine: recent developments in the area of targeted covalent inhibition.
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DOI: 10.1016/j.cbpa.2018.05.011
Abstract: Over the past decade targeted covalent inhibitors have undergone a renaissance due to the clinical validation and regulatory approval of several small molecule therapeutics that are designed to irreversibly modify their target protein. Invariably, these… read more here.
Keywords: beyond cysteine; targeted covalent; area targeted; cysteine recent ... See more keywords