Catalytic Approaches to Optically Active 1,5-Benzothiazepines
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DOI: 10.1021/acscatal.8b00908
Abstract: The 1,5-benzothiazepine framework is well-known as a versatile pharmacophore, and its derivatives have numerous biological activities. Therefore, various synthetic routes to these important compounds have already been investigated. However, in light of the increase in… read more here.
Keywords: optically active; catalytic approaches; benzothiazepine; active benzothiazepines ... See more keywords
Evaluation of 2,3-Dihydro-1,5-benzothiazepine Derivatives as Potential Tyrosinase Inhibitors: In Vitro and In Silico Studies
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DOI: 10.1021/acsomega.3c01566
Abstract: Benzothiazepines are pharmacologically active compounds, frequently utilized as a precursor for acquiring versatile molecules with several bioactivities including anti-inflammatory, anti-human immunodeficiency virus (anti-HIV), analgesic, antitumor, antimicrobial, and antitubercular. In this study, the 2,4-diphenyl-2,3-dihydro-1,5-benzothiazepine scaffold was… read more here.
Keywords: silico studies; dihydro benzothiazepine; benzothiazepine; tyrosinase inhibitors ... See more keywords