Articles with "bioavailability absorption" as a keyword



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A Phase 1 Study to Evaluate Absolute Bioavailability and Absorption, Distribution, Metabolism, and Excretion of Savolitinib in Healthy Male Volunteers

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Published in 2023 at "Clinical Pharmacology in Drug Development"

DOI: 10.1002/cpdd.1224

Abstract: Savolitinib is an oral MET (hepatocyte growth factor receptor) tyrosine kinase inhibitor, with demonstrated preliminary efficacy in several cancer types. Previous pharmacokinetics assessments showed that savolitinib is rapidly absorbed but there are limited data on… read more here.

Keywords: metabolism; bioavailability; savolitinib; bioavailability absorption ... See more keywords