The AMPA receptor biophysical gating properties and binding site: Focus on novel curcumin-based diazepines as non-competitive antagonists.
Sign Up to like & getrecommendations! Published in 2021 at "Bioorganic chemistry"
DOI: 10.1016/j.bioorg.2021.105406
Abstract: INTRODUCTION Investigating the binding site of six novel curcumin-based diazepine compounds as a non-competitive antagonist on ionotropic, AMPA-type glutamate receptors, including homomeric and heteromeric subunits. These receptors play a pivotal role in neurodegenerative diseases such… read more here.
Keywords: binding site; non competitive; biophysical gating; curcumin based ... See more keywords
Effect of Geraniol and Citronellol Essential Oils on the Biophysical Gating Properties of AMPA Receptors
Sign Up to like & getrecommendations! Published in 2019 at "Applied Sciences"
DOI: 10.3390/app9214693
Abstract: Essential oils have been advertised endlessly to be very beneficial for the health of humans, and an extensive amount of research examines the validity of such claims. In contribution, the current study evaluates the neuroprotective… read more here.
Keywords: gating properties; effect; biophysical gating; desensitization deactivation ... See more keywords