SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K.
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DOI: 10.1021/acsmedchemlett.9b00399
Abstract: Inhibitors based on a 3-acylaminoindazole scaffold were synthesized to yield potent dual AAK1/BMP2K inhibitors. Optimization furnished a small molecule chemical probe (SGC-AAK1-1, 25) that is potent and selective for AAK1/BMP2K over other NAK family members,… read more here.
Keywords: aak1 bmp2k; sgc aak1; bmp2k; chemical probe ... See more keywords