Extending the γ-class carbonic anhydrases inhibition profiles with phenolic compounds.
Sign Up to like & getrecommendations! Published in 2019 at "Bioorganic chemistry"
DOI: 10.1016/j.bioorg.2019.103336
Abstract: γ-Class carbonic anhydrases (CAs; EC 4.2.1.1) lack of extended inhibition characterization in comparison to α- and β-class isozymes. For this reason, a panel of 22 phenols was investigated here for the inhibition of the γ-CAs… read more here.
Keywords: class; carbonic anhydrases; inhibition; extending class ... See more keywords
Activation of α-, β-, γ- δ-, ζ- and η- class of carbonic anhydrases with amines and amino acids: a review
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DOI: 10.1080/14756366.2019.1664501
Abstract: Abstract Eight genetically distinct carbonic anhydrase (EC 4.2.1.1) enzyme families (α-, β-, γ- δ-, ζ-, η-, θ- and ι-CAs) were described to date. On the other hand, 16 mammalian α-CA isoforms are known to be… read more here.
Keywords: amino acids; amines amino; carbonic anhydrases; class carbonic ... See more keywords
Anion Inhibition Studies of the β-Class Carbonic Anhydrase CAS3 from the Filamentous Ascomycete Sordaria macrospora
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DOI: 10.3390/metabo10030093
Abstract: CAS3 is a newly cloned cytosolic β-class carbonic anhydrase (CA, EC 4.2.1.1) from the filamentous ascomycete Sordaria macrospora. This enzyme has a high catalytic activity for the physiological CO2 hydration reaction and herein, we report… read more here.
Keywords: carbonic anhydrase; inhibition; ascomycete sordaria; class carbonic ... See more keywords