Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSD1 activity
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DOI: 10.1080/14756366.2022.2052869
Abstract: Abstract As regioisomers/bioisosteres of 1a, a 4-phenylbenzamide tranylcypromine (TCP) derivative previously disclosed by us, we report here the synthesis and biological evaluation of some (hetero)arylbenzoylamino TCP derivatives 1b-6, in which the 4-phenyl moiety of 1a… read more here.
Keywords: derivatives endowed; containing tranylcypromine; heterocycle containing; endowed high ... See more keywords