Design, synthesis, and biological evaluation of pleuromutilin derivatives containing 1,2,4-triazole linker.
Sign Up to like & getrecommendations! Published in 2023 at "Drug development research"
DOI: 10.1002/ddr.22050
Abstract: A series of thioether pleuromutilin derivatives containing 1,2,4‐triazole on the side chain of C14 were designed and synthesized. The in vitro antibacterial activities experiments of the synthesized derivatives showed that compounds 72 and 73 displayed… read more here.
Keywords: design synthesis; synthesis biological; containing triazole; pleuromutilin derivatives ... See more keywords
Design, Synthesis, and Antifungal Evaluation of Novel Benzoxazole Derivatives Containing a 1,2,3‐Triazole Moiety
Sign Up to like & getrecommendations! Published in 2017 at "Journal of The Chinese Chemical Society"
DOI: 10.1002/jccs.201700129
Abstract: For finding novel bioactive compounds with significant antifungal activities, 17 novel benzoxazole derivatives containing a 1,2,3-triazole moiety were synthesized by the copper(II) acetylacetonate-catalyzed cyclization reaction between 2-aminophenol derivatives and 1H-1,2,3-triazole-4-carbaldehyde derivatives (4a), which were prepared… read more here.
Keywords: novel benzoxazole; containing triazole; triazole moiety; benzoxazole derivatives ... See more keywords
Synthesis, in vitro urease inhibition and molecular docking studies of some novel quinazolin-4(3H)-one derivatives containing triazole, thiadiazole and thiosemicarbazide functionalities.
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DOI: 10.1016/j.bioorg.2018.10.031
Abstract: A new series of quinazolinone derivatives containing triazole, thiadiazole, thiosemicarbazide functionalities was synthesized and then screened for their in vitro urease inhibition properties. Most of the compounds showed excellent activity with IC50 values ranging between… read more here.
Keywords: thiosemicarbazide functionalities; vitro urease; thiadiazole thiosemicarbazide; containing triazole ... See more keywords
Preparation of bridged polysilsesquioxane-based membranes containing 1,2,3-triazole moieties for water desalination
Sign Up to like & getrecommendations! Published in 2017 at "Polymer Journal"
DOI: 10.1038/pj.2016.128
Abstract: New organically bridged trialkoxysilanes containing 1,2,3-triazole moieties were synthesized. They were polymerized by sol–gel reactions, giving bridged silica membranes. Water separation properties of the membrane were investigated using a 2000 p.p.m. NaCl aqueous solution, as being… read more here.
Keywords: polysilsesquioxane based; containing triazole; water; bridged polysilsesquioxane ... See more keywords