Deaminative Cyclization of Tertiary Amines for the Synthesis of 2-Arylquinoline Derivatives with a Nonsubstituted Vinylene Fragment.
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DOI: 10.1021/acs.orglett.2c03904
Abstract: With triethylamine as a vinylene source, a convenient protocol for the regioselective synthesis of β,γ-nonsubstituted 2-arylquinolines from aldehydes and arylamines has been accomplished. The deaminative cyclization is also extended to long-chain tertiary alkylamines, enabling diverse… read more here.
Keywords: cyclization tertiary; deaminative cyclization; amines synthesis; tertiary amines ... See more keywords