Shape linear peptides into rigid rings: a sp3 C–H arylation approach to cyclophane-braced peptide macrocycles
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DOI: 10.1007/s11426-018-9288-2
Abstract: Peptide-based therapeutics have attracted increasing attention due to their unique properties in comparison to small molecule drugs and recombinant biologics [1]. With moderate size and suitable surface area, peptides possess enormous potential in drug discovery… read more here.
Keywords: cyclophane braced; peptide macrocycles; braced peptide; arylation ... See more keywords