Size-Dependent Target Engagement of Covalent Probes
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DOI: 10.1021/acs.jmedchem.5c00017
Abstract: Labeling proteins with covalent ligands is finding increasing use in proteomics applications, including identifying nucleophilic residues amenable for labeling and in the development of targeted covalent inhibitors (TCIs). Labeling efficiency is measured by the covalent… read more here.
Keywords: covalent; dependent target; size dependent; target engagement ... See more keywords