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Published in 2017 at "Future medicinal chemistry"
DOI: 10.4155/fmc-2017-0074
Abstract: AIM DNA methyltransferases (DNMTs) are important drug targets for epigenetic therapy of cancer. Nowadays, non-nucleoside DNMT inhibitors are in development to address high toxicity of nucleoside analogs. However, these compounds still have low activity in…
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Keywords:
maleimide derivatives;
inhibition studies;
dna methyltransferases;
non nucleoside ... See more keywords