Development of a sp2-sp3 Stille Cross-Coupling for Rapid Synthesis of HIV NNRTI Doravirine Analogues.
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DOI: 10.1021/acs.orglett.7b01142
Abstract: The development of a C(sp2)-C(sp3) cross-coupling reaction for rapid, parallel synthesis of analogues of two HIV NNRTI clinical candidates is described. This method allowed easy access to the C-ring space using a practical alkylation with… read more here.
Keywords: sp2 sp3; development sp2; hiv nnrti; cross coupling ... See more keywords