A facile and efficient synthesis of 3‐cyanoindoles by a simple palladium(II)‐catalyzed C─H activation of indoles
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DOI: 10.1002/aoc.3706
Abstract: An efficient trans-PdCl2(NH2CH2COOH)2-catalyzed direct C3-cyanation of indole C─H bonds is described. Notably, free (N─H)-indoles reacted smoothly using the procedure, and the desired product 3-cyanoindoles were obtained in good to excellent yields. read more here.
Keywords: simple palladium; efficient synthesis; facile efficient; palladium catalyzed ... See more keywords
Green and efficient synthesis of an adsorbent fiber by preirradiation‐induced grafting of PDMAEMA and its Au(III) adsorption and reduction performance
Sign Up to like & getrecommendations! Published in 2017 at "Journal of Applied Polymer Science"
DOI: 10.1002/app.44955
Abstract: N,N-Dimethylamino ethyl methacrylate (DMAEMA) is covalently bonded on a commercial polyethylene-coated polypropylene skin-core structure fiber (PE/PP) in aqueous and MeOH/H2O solutions by a one-step green reaction using radiation-induced graft polymerization. The effects of the absorbed… read more here.
Keywords: adsorption; synthesis adsorbent; adsorbent fiber; efficient synthesis ... See more keywords
Efficient Synthesis of Cleavable Cell‐Penetrating Peptide–Cargo Conjugate via Low‐Equivalent of Cell‐Penetrating Peptide Activated by 2,2′‐Dithiodipyridine
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DOI: 10.1002/cbic.202500032
Abstract: Cell‐penetrating peptides (CPPs) are favored for protein delivery due to their efficiency, rapidity, and low toxicity. However, conjugation of CPPs to proteins often requires significant amounts of CPPs to ensure yields, which also may result… read more here.
Keywords: cargo; synthesis cleavable; penetrating peptide; cell ... See more keywords
Enzyme‐Catalyzed Efficient Synthesis of Enantiomerically Pure (S)‐ and (R)‐n‐Butylphthalide
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DOI: 10.1002/cbic.202500482
Abstract: 3‐n‐Butylphthalide (NBP) is an effective commercial drug for the treatment of acute ischemic stroke, with its S‐enantiomer, (S)‐NBP, demonstrating clinical superiority over (R)‐NBP. However, the stereoselective synthesis of both enantiomers with high enantiomeric excess (ee)… read more here.
Keywords: enantiomerically pure; catalyzed efficient; synthesis; enzyme catalyzed ... See more keywords
An Efficient Synthesis of 3‐Alkylpyridine Alkaloids Enables Their Biological Evaluation
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DOI: 10.1002/cmdc.202100134
Abstract: 3‐Alkylpyridine alkaloids (3‐APAs) isolated from the arctic sponge Haliclona viscosa are a promising group of bioactive marine alkaloids. However, due to limited bioavailability, investigations of their bioactivity have been hampered. Additionally, synthesis of a common… read more here.
Keywords: biological evaluation; alkylpyridine alkaloids; efficient synthesis; alkaloids enables ... See more keywords
Efficient Synthesis of Cyclic Carbonates from Unsaturated Acids and Carbon Dioxide and their Application in the Synthesis of Biobased Polyurethanes.
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DOI: 10.1002/cplu.202100079
Abstract: Bio-derived furan- and diacid-derived cyclic carbonates have been synthesized in high yields from terminal epoxides and CO2 . Furthermore, four highly substituted terpene-derived cyclic carbonates were isolated in good yields with excellent diastereoselectivity in some… read more here.
Keywords: synthesis cyclic; efficient synthesis; unsaturated acids; carbonates unsaturated ... See more keywords
Mild and Efficient Synthesis of Diverse Organo‐AuI‐L Complexes in Green Solvents
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DOI: 10.1002/cssc.201903415
Abstract: Abstract An exceptionally mild and efficient method was developed for the preparation of (hetero)aryl‐AuI‐L complexes using ethanol or water as the reaction medium at room temperature and Ar‐B(triol)K boronates as the transmetalation partner. The reaction… read more here.
Keywords: efficient synthesis; reaction; aryl; mild efficient ... See more keywords
A Mild and Efficient Synthesis of Functionalized 2‐Fluorobenzamides from 1,2,3‐Benzotriazinones via Denitrogenative Fluorination Reactions under Thermal/Visible Light Conditions
Sign Up to like & getrecommendations! Published in 2025 at "European Journal of Organic Chemistry"
DOI: 10.1002/ejoc.202500375
Abstract: An efficient method for the synthesis of 2‐fluorobenzamides was established from 1,2,3‐benzotriazinones using tetrafluoroboric acid. The reactions proceeded under mild thermal conditions, providing a wide range of functionalized 2‐fluorobenzamides in 65‐80% yields. On the other… read more here.
Keywords: functionalized fluorobenzamides; mild efficient; visible light; synthesis functionalized ... See more keywords
An Efficient Synthesis of 6′‐methyl‐1'H‐spiro[indoline‐3,4′‐pyrimidine]‐2,2′(3'H)‐dione Derivatives
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DOI: 10.1002/jhet.2944
Abstract: The reactions of isatins, urea and 1-(piperidin-1-yl)butane-1,3-dione or 1-morpholinobutane-1,3-dione have been developed for the preparation of spiroheterocycles compounds. It was found these reactions could be given higher yields and required shorter time in our process.… read more here.
Keywords: dione; efficient synthesis; methyl spiro; spiro indoline ... See more keywords
An Efficient Synthesis and Antibacterial Activity of Some Novel 2-Azetidinone Derivatives of 4H-1,2,4-Triazoles Under Mild Conditions
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DOI: 10.1002/jhet.3136
Abstract: We have synthesized the novel 2-azetidinone derivatives by using Schiff bases of 1,2,4-triazoles via a single step protocol. We used DABCO as a good homogenous, ecofriendly, highly reactive, easy to handle, and nontoxic catalyst. In DABCO… read more here.
Keywords: efficient synthesis; azetidinone derivatives; synthesis antibacterial; novel azetidinone ... See more keywords
Efficient Synthesis of 1‐Chloroimidazo[1,2‐a:4,5‐c']dipyridines, Versatile Synthons for Position‐1 Functionalisation with Various Reagents
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DOI: 10.1002/open.202500178
Abstract: In this work, the goal is to develop a versatile synthetic pathway to functionalize position‐1 of the imidazo[1,2‐a;4,5‐c']dipyridine core. For this purpose, the synthesis of 1‐chloroimidazo[1,2‐a;4,5‐c']dipyridines via a novel synthetic pathway starting from imidazo[1,2‐a]pyridines conveniently… read more here.
Keywords: efficient synthesis; chloroimidazo dipyridines; synthesis chloroimidazo; position ... See more keywords