PIDA‐Enabled C3‐Amination of Imidazopyridines with Primary Aromatic Amines Using Rongalite as In Situ C1 Source
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DOI: 10.1002/ajoc.70189
Abstract: Imidazo[1,2‐a]pyridine represents a significant heterocyclic scaffold, and its C3‐aminated derivatives demonstrate enhanced bioactivity. However, employing primary arylamines directly as aminating agents remains challenging to date. Herein, we report the PIDA‐enabled C3‐amination of imidazopyridines employing primary… read more here.
Keywords: enabled amination; aromatic amines; primary aromatic; amination ... See more keywords