Articles with "enantiomers human" as a keyword



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Comparative metabolism and tolerability of racemic primaquine and its enantiomers in human volunteers during 7-day administration

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Published in 2023 at "Frontiers in Pharmacology"

DOI: 10.3389/fphar.2022.1104735

Abstract: Primaquine (PQ) is an 8-aminoquinoline antimalarial, active against dormant Plasmodium vivax hypnozoites and P. falciparum mature gametocytes. PQ is currently used for P. vivax radical cure and prevention of malaria transmission. PQ is a racemic… read more here.

Keywords: primaquine; metabolism; pharmacology; tolerability ... See more keywords