Copper-catalyzed asymmetric dearomative borylation: new pathway to optically active heterocyclic compounds
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DOI: 10.1515/pac-2017-0912
Abstract: Abstract Chiral N-heterocyclic organoboronates represent promising intermediates for the preparation of various bioactive and pharmaceutical compounds. We recently reported the first asymmetric dearomative borylation of indoles by copper-catalyzed borylation. Then we further developed dearomatization/enantioselective borylation… read more here.
Keywords: enantioselective borylation; borylation; asymmetric dearomative; dearomative borylation ... See more keywords