Articles with "formulations strategic" as a keyword



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Liposome Formulations for the Strategic Delivery of PARP1 Inhibitors: Development and Optimization

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Published in 2023 at "Nanomaterials"

DOI: 10.3390/nano13101613

Abstract: The development of a lipid nano-delivery system was attempted for three specific poly (ADP-ribose) polymerase 1 (PARP1) inhibitors: Veliparib, Rucaparib, and Niraparib. Simple lipid and dual lipid formulations with 1,2-dipalmitoyl-sn-glycero-3-phospho-rac-(1′-glycerol) sodium salt (DPPG) and 1,2-dipalmitoyl-sn-glycero-3-phosphocoline… read more here.

Keywords: formulations strategic; parp1 inhibitors; development; liposome formulations ... See more keywords