Rigid H4OCTAPA derivatives as model chelators for the development of Bi(III)-based radiopharmaceuticals.
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DOI: 10.1039/d2cc06876a
Abstract: Octadentate ligands containing ethyl (H4OCTAPA), cyclohexyl (H4CHXOCTAPA) or cyclopentyl (H4CpOCTAPA) spacers were assessed as chelators for Bi(III)-based radiopharmaceuticals. The H4CHXOCTAPA chelator displays excellent properties, including 205/206Bi-nuclide radiolabelling under mild conditions, excellent stability in serum and… read more here.
Keywords: h4octapa derivatives; derivatives model; based radiopharmaceuticals; iii based ... See more keywords