Articles with "inhibitors degraders" as a keyword



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Targeting Brd4 for cancer therapy: inhibitors and degraders.

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Published in 2018 at "MedChemComm"

DOI: 10.1039/c8md00198g

Abstract: Bromodomain-containing protein 4 (Brd4) plays an important role in mediating the expression of genes involved in cancers and non-cancer diseases such as inflammatory diseases and acute heart failure. Inactivating Brd4 or downregulating its expression inhibits… read more here.

Keywords: targeting brd4; brd4 cancer; brd4; cancer ... See more keywords