A Fast Track to Indoles and Annulated Indoles through ortho- vs ipso-Amination of Aryl Halides.
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DOI: 10.1021/acs.orglett.9b04202
Abstract: A complementary site selective ortho- vs ipso-amination of aryl halides using non-electrophilic amine sources for construction of indole scaffolds is reported. A palladium-catalyzed alkyne insertion/C-H activation/palladacycle amination via merger of three easily diversified components including… read more here.
Keywords: ipso amination; amination; aryl halides; amination aryl ... See more keywords