An Integrated Approach toward NanoBRET Tracers for Analysis of GPCR Ligand Engagement
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DOI: 10.3390/molecules26102857
Abstract: Gaining insight into the pharmacology of ligand engagement with G-protein coupled receptors (GPCRs) under biologically relevant conditions is vital to both drug discovery and basic research. NanoLuc-based bioluminescence resonance energy transfer (NanoBRET) monitoring competitive binding… read more here.
Keywords: ligand engagement; ligand; fluorescent tracers; approach ... See more keywords