Palladium-Catalyzed Oxidation-Hydroxylation and Oxidation-Methoxylation of N-Boc Indoles for the Synthesis of 3-Oxoindolines
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DOI: 10.1055/s-0036-1589032
Abstract: The palladium-catalyzed oxidation-hydroxylation and oxidation-methoxylation of N-Boc indoles for the synthesis of tert-butyl 2-hydroxy(methoxy)-3-oxoindoline-1-carboxylates and their derivatives is developed. The process occurs readily using PdCl2 as the catalyst and acetonitrile as the solvent to afford… read more here.
Keywords: hydroxylation oxidation; oxidation; oxidation hydroxylation; methoxylation boc ... See more keywords