Extended Applications of Small-Molecule Covalent Inhibitors toward Novel Therapeutic Targets
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DOI: 10.3390/ph15121478
Abstract: Recently, small-molecule covalent inhibitors have been accepted as a practical tool for targeting previously “undruggable” proteins. The high target selectivity of modern covalent inhibitors is now alleviating toxicity concerns regarding the covalent modifications of proteins.… read more here.
Keywords: small molecule; covalent inhibitors; molecule covalent; extended applications ... See more keywords