Native Amino Group Directed Site-Selective ε-C(sp2)-H Iodination of Primary Amines.
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DOI: 10.1021/acs.orglett.2c04288
Abstract: Selective remote C-H activating amines using unmodified NH2 as a native directing group demonstrate compelling synthetic utilities. The 3-arylpropan-1-amine moiety is present in many drugs and candidates in clinical trials. Selective iodination of 3-arylpropan-1-amines on… read more here.
Keywords: native amino; sp2 iodination; selective sp2; group ... See more keywords