Novel Aryl Boronate Ester Based Amino Acids as Orthogonal Building Blocks for Fmoc Solid Phase Peptide Synthesis
Sign Up to like & getrecommendations! Published in 2017 at "European Journal of Organic Chemistry"
DOI: 10.1002/ejoc.201701064
Abstract: Three novel aryl boronate ester based amino acids are described. These useful building blocks were found to exhibit all of the chemical properties compatible to the Fmoc strategy solid-phase peptide synthesis and orthogonal to Boc,… read more here.
Keywords: novel aryl; solid phase; peptide synthesis; phase peptide ... See more keywords
Discovery of novel (N-aryl-4-methylpiperidinyl)pyrazoles: A new class of potent lepidopteran insecticides.
Sign Up to like & getrecommendations! Published in 2023 at "Pest management science"
DOI: 10.1002/ps.7349
Abstract: BACKGROUND Insects of the order Lepidoptera are among the most destructive global pests causing billions of dollars in damage annually. A new class of N-arylpyrazole-4-methylpiperidines with potent activity on lepidopteran species has been discovered. RESULTS… read more here.
Keywords: discovery novel; novel aryl; class; new class ... See more keywords
Discovery of novel 2-aryl-3-sulfonamido-pyridines (HoAns) as microtubule polymerization inhibitors with potent antitumor activities.
Sign Up to like & getrecommendations! Published in 2020 at "European journal of medicinal chemistry"
DOI: 10.1016/j.ejmech.2020.113117
Abstract: Microtubules play a vital role in cell mitosis. Drugs targeting taxol or vinca binding site of tubulin have been proved an effective way to against cancer. However, drug resistance and cancer recurrence are inevitable, there… read more here.
Keywords: aryl sulfonamido; novel aryl; pyridines hoans; compound hoan32 ... See more keywords
Design, Synthesis, and Structure-Activity Relationship of Novel Aryl-Substituted Formyl Oxazolidine Derivatives as Herbicide Safeners.
Sign Up to like & getrecommendations! Published in 2023 at "Journal of agricultural and food chemistry"
DOI: 10.1021/acs.jafc.3c00467
Abstract: Nicosulfuron is the leading herbicide in the global sulfonylurea (SU) herbicide market; it was jointly developed by DuPont and Ishihara. Recently, the widespread use of nicosulfuron has led to increasingly prominent agricultural production hazards, such… read more here.
Keywords: compound; structure; novel aryl; herbicide safeners ... See more keywords
Synthesis and Characterization of Novel 4-aryl-4H-chromene Derivatives Using Borax and Evaluation of their Anticancer Effects.
Sign Up to like & getrecommendations! Published in 2023 at "Anti-cancer agents in medicinal chemistry"
DOI: 10.2174/1871520623666230504101651
Abstract: 4-aryl-4H-chromenes have attracted attention as potential anticancer agents. In an effort to discover effective compounds, we designed a new series of these chromenes with methoxy substitution at 2, 3, 4, 5, and 6 positions. The… read more here.
Keywords: characterization novel; cell; novel aryl; cell line ... See more keywords