Discovery of b-Arrestin Biased, Orally Bioavailable and CNS Penetrant Neurotensin Receptor 1 (NTR1) Allosteric Modulators.
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DOI: 10.1021/acs.jmedchem.9b00340
Abstract: Neurotensin receptor 1 (NTR1) is a G protein coupled receptor that is widely expressed throughout the central nervous sys-tem where it acts as a neuromodulator. Neurotensin receptors have been implicated in a wide variety of… read more here.
Keywords: neurotensin receptor; receptor ntr1; cns; ntr1 allosteric ... See more keywords