Ethyl Pinacol Boronates as Advantageous Precursors for Copper-Mediated Radiofluorination
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DOI: 10.1021/acs.orglett.5c02055
Abstract: (Hetero)aryl pinacol boronic esters are routinely used for 18F-labeling and have accelerated numerous diagnostic and drug discovery programs. An analysis of the current state-of-play, however, highlights a pending challenge. Reports have indicated that some pinacol… read more here.
Keywords: copper mediated; pinacol; pinacol boronates; boronic esters ... See more keywords