Edmond Fischer's kinase legacy: History of the protein kinase inhibitor and protein kinase A
Sign Up to like & getrecommendations! Published in 2023 at "IUBMB Life"
DOI: 10.1002/iub.2714
Abstract: Although Fischer's extraordinary career came to focus mostly on the protein phosphatases, after his co‐discovery of Phosphorylase Kinase with Ed Krebs he was clearly intrigued not only by cAMP‐dependent protein kinase (PKA), but also by… read more here.
Keywords: protein kinase; pka; pki; inhibitor ... See more keywords
A Non-imaging High Throughput Approach to Chemical Library Screening at the Unmodified Adenosine-A3 Receptor in Living Cells
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DOI: 10.3389/fphar.2017.00908
Abstract: Recent advances in fluorescent ligand technology have enabled the study of G protein-coupled receptors in their native environment without the need for genetic modification such as addition of N-terminal fluorescent or bioluminescent tags. Here, we… read more here.
Keywords: affinity; non imaging; adenosine receptor; plate ... See more keywords