Biological evaluation of some quinoline derivatives with different functional groups as anticancer agents
Sign Up to like & getrecommendations! Published in 2019 at "Journal of Biochemical and Molecular Toxicology"
DOI: 10.1002/jbt.22260
Abstract: Due to a great deal of biological activities, quinoline derivatives have drawn attention for synthesis and biological activities in the search for new anticancer drug development. In this work, a variety of substituted (phenyl, nitro,… read more here.
Keywords: biological evaluation; evaluation quinoline; bromo nitroquinoline; activity ... See more keywords
Theoretical-Experimental Photophysical Investigations of the Solvent Effect on the Properties of Green- and Blue-Light-Emitting Quinoline Derivatives
Sign Up to like & getrecommendations! Published in 2017 at "Journal of Fluorescence"
DOI: 10.1007/s10895-017-2108-0
Abstract: This paper describes the investigations on the solvatochromic effect and the photophysical properties of quinoline derivatives, compounds with potential applicability in optoelectronic devices. Using an experimental and theoretical approach, the effect of the solvent and… read more here.
Keywords: photophysical investigations; theoretical experimental; experimental photophysical; effect ... See more keywords
Microwave-irradiated one-pot synthesis of quinoline derivatives catalyzed by triethylamine
Sign Up to like & getrecommendations! Published in 2017 at "Research on Chemical Intermediates"
DOI: 10.1007/s11164-017-2986-4
Abstract: An efficient and swift microwave (MW)-mediated procedure for synthesis of 11 quinoline derivatives has been designed based on reaction between aromatic aldehydes, malononitrile, 5,5-dimethylcyclohexane-1,3-dione, and ammonium acetate at room temperature in ethanol solvent. The main… read more here.
Keywords: synthesis quinoline; microwave irradiated; irradiated one; quinoline derivatives ... See more keywords
Copper catalyzed oxidative coupling of ortho-vinylanilines with N-tosylhydrazones: Efficient synthesis of polysubstituted quinoline derivatives
Sign Up to like & getrecommendations! Published in 2018 at "Journal of Catalysis"
DOI: 10.1016/j.jcat.2018.04.005
Abstract: Abstract Efficient and general copper catalyzed oxidative cyclization of ortho-vinylaniline has been accomplished employing N-tosylhydrazone as coupling partner. Various substituted quinoline derivatives of biological importance were achieved in good to excellent yield. The important features… read more here.
Keywords: copper catalyzed; quinoline derivatives; coupling ortho; oxidative coupling ... See more keywords
Structural Simplification of Cryptolepine to Obtain Novel Antifungal Quinoline Derivatives against Phytopathogenic Fungi.
Sign Up to like & getrecommendations! Published in 2023 at "Journal of agricultural and food chemistry"
DOI: 10.1021/acs.jafc.2c07575
Abstract: A series of quinoline derivatives were designed and synthesized by the structural simplification of cryptolepine and evaluated for their fungicidal activity against six phytopathogenic fungi. Most of these compounds exhibited remarkable activities against Botrytis cinereain… read more here.
Keywords: quinoline derivatives; cryptolepine; structural simplification; compound a18 ... See more keywords
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening.
Sign Up to like & getrecommendations! Published in 2022 at "ACS medicinal chemistry letters"
DOI: 10.1021/acsmedchemlett.2c00249
Abstract: A virtual screening approach based on a five-feature pharmacophoric model for negative modulators of GLI1 was applied to databases of commercially available compounds. The resulting quinoline derivatives showed significant ability to reduce the GLI1 protein… read more here.
Keywords: quinoline derivatives; quinolines oxazino; derivatives small; virtual screening ... See more keywords
Facile Route to the Synthesis of 1,3-Diazahetero-Cycle-Fused [1,2-a]Quinoline Derivatives via Cascade Reactions
Sign Up to like & getrecommendations! Published in 2018 at "ACS Omega"
DOI: 10.1021/acsomega.7b01856
Abstract: A one-step protocol without transition-metal catalysts with simple post-treatment for the synthesis of 1,3-diazaheterocycle-fused [1,2-a]quinoline derivatives via the cascade reaction of 2-fluorobenzaldehyde (1) and heterocyclic ketene aminals (2) was developed. In the one-step cascade reaction,… read more here.
Keywords: via cascade; facile route; fused quinoline; derivatives via ... See more keywords
Zircon PrVO4: an efficient heterogeneous catalyst for tandem oxidative synthesis of 2,3-disubstituted quinoline derivatives.
Sign Up to like & getrecommendations! Published in 2023 at "Dalton transactions"
DOI: 10.1039/d3dt00435j
Abstract: The current study addresses the usage of inherent redox couplets in PrVO4 crystallizing in a zircon-type structure for tandem oxidative transformation. Monophasic PrVO4, synthesized using a solution combustion synthesis method, showed a tetragonal zircon-type structure… read more here.
Keywords: synthesis disubstituted; quinoline derivatives; synthesis; zircon prvo4 ... See more keywords
Recent reviews on quinoline derivatives as corrosion inhibitors
Sign Up to like & getrecommendations! Published in 2018 at "Corrosion Reviews"
DOI: 10.1515/corrrev-2017-0129
Abstract: Abstract Traditionally, controlling corrosion has been managed by various methods like cathodic protection, process control, reduction of the metal impurity content and application of surface treatment techniques as well as incorporation of suitable alloys. However,… read more here.
Keywords: derivatives corrosion; corrosion inhibitors; quinoline derivatives; reviews quinoline ... See more keywords
Antioxidant effect of quinoline derivatives containing or not selenium: Relationship with antinociceptive action quinolines are antioxidant and antinociceptive.
Sign Up to like & getrecommendations! Published in 2017 at "Anais da Academia Brasileira de Ciencias"
DOI: 10.1590/0001-3765201720160668
Abstract: The present study investigated the antioxidant effect of a new class of quinoline derivatives (a-d) on assays in vitro. Lipid peroxidation, thiol peroxidase-like and free radical scavenging activities were determined to evaluate antioxidant activity of… read more here.
Keywords: antioxidant effect; lipid peroxidation; effect; compound ... See more keywords
Synthesis of Fused Quinoline Derivatives With Antiproliferative Activities and Tyrosine Kinases, Pim-1 Kinase Inhibitions.
Sign Up to like & getrecommendations! Published in 2022 at "Acta chimica Slovenica"
DOI: 10.17344/acsi.2021.6733
Abstract: Cyclohexan-1,3-dione (1) reacted with either 2-aminoprop-1-ene-1,1,3-tricarbonitrile (2a) or diethyl 3-amino-2-cyanopent-2-enedioate (2b) to give the 5,6,7,8-tetrahydronaphthalene derivatives 3a and 3b, respectively. The latter compounds underwent further heterocyclization reactions to give the thieno[2',3':5,6]benzo[1,2-e][1,3]oxazine derivatives. On the other… read more here.
Keywords: quinoline derivatives; derivatives antiproliferative; tyrosine kinases; synthesis fused ... See more keywords