The regioselective coupling of 2-arylquinazolinone C–H with aldehydes and benzyl alcohols under oxidative conditions
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DOI: 10.1039/d0nj03721d
Abstract: The direct and regioselective palladium-catalyzed dehydrogenative coupling of aldehydes and benzyl alcohols with 2-aryl-quinazolinone C–H endowed with a quinazolinone nucleus, which is one of the most fascinating and vital core units, as an inherent directing… read more here.
Keywords: oxidative conditions; regioselective coupling; aldehydes benzyl; coupling arylquinazolinone ... See more keywords
Palladium-Catalyzed Regioselective Coupling of Secondary Propargyl Carbonates and Ethyl 2-(pyridin-2-yl)acetate Derivatives: Facile Access to C-3 Benzylated Indolizines
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DOI: 10.1055/s-0037-1609552
Abstract: A palladium-catalyzed ligand controlled regioselective coupling reaction of secondary propargyl carbonates and ethyl 2-(pyridin-2-yl)acetate derivatives has been described, leading to C-3 benzylated indolizines for the first time in moderate to good yields. DBFphos as the… read more here.
Keywords: regioselective coupling; secondary propargyl; palladium catalyzed; carbonates ethyl ... See more keywords