Structure–Activity Relationships of 1‐Benzoylazulenes at the OX1 and OX2 Orexin Receptors
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DOI: 10.1002/cmdc.201900074
Abstract: We previously demonstrated the potential of di‐ or trisubstituted azulenes as ligands (potentiators, weak agonists, and antagonists) of the orexin receptors. In this study we investigated 27 1‐benzoylazulene derivatives, uncovering seven potentiators of the orexin… read more here.
Keywords: orexin receptors; activity relationships; relationships benzoylazulenes; structure activity ... See more keywords