Peptide stapling by late-stage Suzuki–Miyaura cross-coupling
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DOI: 10.3762/bjoc.18.1
Abstract: The development of peptide stapling techniques to stabilise α-helical secondary structure motifs of peptides led to the design of modulators of protein–protein interactions, which had been considered undruggable for a long time. We disclose a… read more here.
Keywords: cross coupling; suzuki miyaura; stage suzuki; peptide stapling ... See more keywords