Peptide Stapling through Site-Directed Conjugation of Triazine Moieties to the Tyrosine Residues of a Peptide.
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DOI: 10.1021/acs.orglett.3c00499
Abstract: Peptide stapling is a strategy for improving the biological properties of peptides. Herein, we report a novel method for stapling peptides that utilizes bifunctional triazine moieties for two-component conjugation to the phenolic hydroxyl groups of… read more here.
Keywords: triazine moieties; conjugation; site directed; peptide stapling ... See more keywords