Discovery of Novel Substrate-Competitive Lysine Methyltransferase G9a Inhibitors as Anticancer Agents.
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DOI: 10.1021/acs.jmedchem.2c02059
Abstract: Identification of structurally novel inhibitors of lysine methyltransferase G9a has been a subject of intense research in cancer epigenetics. Starting with the high-throughput screening (HTS) hit rac-10a obtained from the chemical library of the University… read more here.
Keywords: substrate competitive; methyltransferase g9a; discovery novel; g9a ... See more keywords