Synthesis of pH-sensitive sulfonamide-based hydrogels with controllable crosslinking density by post thermo-curing
Sign Up to like & getrecommendations! Published in 2019 at "Journal of Polymer Research"
DOI: 10.1007/s10965-018-1672-6
Abstract: Sulfonamide-containing linear copolymers were synthesized via copolymerization of N-(4-methacrylamido)-N′-(4,6-dimethylpyrimidin-2-yl) benzene-1-sulfonamide (SAM) and N,N′-dimethylacrylamide (DMAAm) via free-radical polymerization at room temperature using redox initiators. The redox-initiated polymerization could undergo nearly complete reaction in which the copolymer… read more here.
Keywords: post thermo; thermo curing; sulfonamide; crosslinking density ... See more keywords
Synthesis of novel dipeptide sulfonamide conjugates with effective carbonic anhydrase I, II, IX, and XII inhibitory properties.
Sign Up to like & getrecommendations! Published in 2018 at "Bioorganic chemistry"
DOI: 10.1016/j.bioorg.2018.08.032
Abstract: Twenty-four novel sulfonamide derivatives incorporating dipeptide tails were synthesized by facile acylation reactions of homosulfanilamide through benzotriazole or dicyclohexyl carbodiimide (DCC) mediated coupling reactions. The carbonic anhydrase (CA, EC 4.2.1.1) inhibitory activity of the new… read more here.
Keywords: carbonic anhydrase; dipeptide; inhibitory properties; xii ... See more keywords
Electrochemical synthesis of new sulfone and sulfonamide derivatives. A green method based on the electrolysis of 2-amino-5-nitrophenol
Sign Up to like & getrecommendations! Published in 2021 at "Electrochimica Acta"
DOI: 10.1016/j.electacta.2021.139223
Abstract: Abstract 2-Amino-5-nitrophenol (ANP) is an electrochemically interesting compound. It has a nitro group that can be reduced independently and also has hydroxyl and an amine functional groups, making the molecule susceptible to oxidation. These features… read more here.
Keywords: amino nitrophenol; process; sulfonamide; synthesis ... See more keywords
CuI nanoparticle-immobilized on a hybrid material composed of IRMOF-3 and a sulfonamide-based porous organic polymer as an efficient nanocatalyst for one-pot synthesis of 2,4-diaryl-quinolines
Sign Up to like & getrecommendations! Published in 2023 at "RSC Advances"
DOI: 10.1039/d3ra01164j
Abstract: As a significant class of synthetic and natural products with multiple biological activities, quinolines are used in medical and electronic devices. In this study, a novel method is presented to synthesize 2,4-diarylquinoline derivatives via a… read more here.
Keywords: organic polymer; one pot; based porous; porous organic ... See more keywords
Synthesis, structure and sulfonamide-sulfonimide tautomerism of sulfonamide-1,2,4-triazine derivatives.
Sign Up to like & getrecommendations! Published in 2022 at "Acta crystallographica. Section C, Structural chemistry"
DOI: 10.1107/s2053229622007781
Abstract: Two new 1,2,4-triazine-containing sulfonamide derivatives, namely, 4-bromo-N-(5,6-diphenyl-2H-1,2,4-triazin-3-ylidene)benzenesulfonamide, C21H15BrN4O4S, 3a, and methyl 2-{[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfamoyl]methyl}benzoate, C24H20N4O4S, 3b, which crystallize in the different sulfonimide and sulfonamide tautomeric forms, respectively, were synthesized and characterized by spectroscopic, X-ray diffraction and theoretical… read more here.
Keywords: synthesis structure; triazine; tautomeric forms; sulfonamide ... See more keywords
Sulfonamide Residues: Honey Quality in the Czech Market
Sign Up to like & getrecommendations! Published in 2018 at "Journal of Food Quality"
DOI: 10.1155/2018/2939207
Abstract: In this study, we determined four sulfonamide compounds (sulfadiazine, sulfadoxine, sulfamethoxazole, and sulfathiazole) in honey marketed in the Czech Republic (Brno). The content of these compounds was monitored in 50 honeys with different botanical and… read more here.
Keywords: quality czech; quality; sulfonamide residues; honey quality ... See more keywords
Magnetic Carbon Microspheres as a Reusable Adsorbent for Sulfonamide Removal from Water
Sign Up to like & getrecommendations! Published in 2017 at "Nanoscale Research Letters"
DOI: 10.1186/s11671-017-2295-2
Abstract: Novel reusable magnetic carbon microspheres (MCMs) were prepared by hydrothermal method with glucose as carbon source and Fe3O4 nanoparticles as magnetic raw materials. And adsorption performance of MCMs for sulfonamide removal from water was investigated… read more here.
Keywords: adsorption; carbon; carbon microspheres; mcms ... See more keywords
Design, synthesis, ADME prediction and pharmacological evaluation of novel benzimidazole-1,2,3-triazole-sulfonamide hybrids as antimicrobial and antiproliferative agents
Sign Up to like & getrecommendations! Published in 2018 at "Chemistry Central Journal"
DOI: 10.1186/s13065-018-0479-1
Abstract: BackgroundNitrogen heterocyclic rings and sulfonamides have attracted attention of several researchers.ResultsA series of regioselective imidazole-based mono- and bis-1,4-disubstituted-1,2,3-triazole-sulfonamide conjugates 4a–f and 6a–f were designed and synthesized. The first step in the synthesis was a regioselective… read more here.
Keywords: antimicrobial antiproliferative; sulfonamide hybrids; evaluation; benzimidazole triazole ... See more keywords
Recent Advances on Biological Active Sulfonamide based Hybrid Compounds Part B: Two-Component Sulfonamide Hybrids.
Sign Up to like & getrecommendations! Published in 2022 at "Current medicinal chemistry"
DOI: 10.2174/0929867329666220722143547
Abstract: Sulfonamide compounds, also known as sulfa drugs, are a significant class of synthetic bacteriostatic antimicrobials and were the primary source of therapy against bacterial infections before the introduction of penicillin in 1941. Hybridization of sulfonamides… read more here.
Keywords: component sulfonamide; sulfonamide; two component; sulfonamide hybrids ... See more keywords
Anticancer Potential of Sulfonamide Moieties via In-Vitro and In-Silico Approaches: Comparative Investigations for Future Drug Development
Sign Up to like & getrecommendations! Published in 2023 at "International Journal of Molecular Sciences"
DOI: 10.3390/ijms24097953
Abstract: Several kinds of anticancer drugs are presently commercially accessible, but low efficacy, solubility, and toxicity have reduced the overall therapeutic indices. Thus, the search for promising anticancer drugs continues. The interactions of numerous essential anticancer… read more here.
Keywords: anticancer drugs; molecular docking; anticancer potential; development ... See more keywords
Discovery of Novel 3,4-Dihydro-2(1H)-Quinolinone Sulfonamide Derivatives as New Tubulin Polymerization Inhibitors with Anti-Cancer Activity
Sign Up to like & getrecommendations! Published in 2022 at "Molecules"
DOI: 10.3390/molecules27051537
Abstract: In this paper, a small series of novel quinoline sulfonamide derivatives was synthesized, and their structure of the target compounds were confirmed by 1H NMR and MS. The screening of the news target compounds’ in… read more here.
Keywords: discovery novel; sulfonamide derivatives; activity; tubulin polymerization ... See more keywords