Synthesis of Benzimidazole-Fused Medium-Sized N,S -Heterocycles via Palladium-Catalyzed Cyclizations
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DOI: 10.1002/ejoc.201801686
Abstract: The synthesis of unprecedented benzimidazole-fused thiazocines, thiazonines, and thiazecines having an exocyclic double bond is reported. The process consists in an 8-, 9-, or 10-exo-dig cyclocarbopalladation followed by reduction. The scope and limitations were established… read more here.
Keywords: medium sized; fused medium; sized heterocycles; synthesis benzimidazole ... See more keywords
Synthesis of Benzimidazole-1,2,4-triazole Derivatives as Potential Antifungal Agents Targeting 14α-Demethylase
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DOI: 10.1021/acsomega.2c07755
Abstract: Invasive fungal infections (IFIs) are increasing as major infectious diseases around the world, and the limited efficacy of existing medications has resulted in substantial morbidity and death in patients due to the lack of effective… read more here.
Keywords: benzimidazole triazole; triazole derivatives; targeting demethylase; synthesis benzimidazole ... See more keywords
CO2 Improved Synthesis of Benzimidazole with the Catalysis of a New Calcium 4-Amino-3-hydroxybenzoate.
Sign Up to like & getrecommendations! Published in 2021 at "Acta chimica Slovenica"
DOI: 10.17344/acsi.2020.6359
Abstract: In this paper, we explored the synthesis of benzimidazole by the reaction of DMF and o-phenylenediamine. In the process of catalyst screening, we found that 4-amino-3-hydroxybenzoic acid, benzoic acid, and benzene-1,3,5-tricarboxylic acid could catalyze the… read more here.
Keywords: co2; amino hydroxybenzoate; calcium amino; amino ... See more keywords
Montmorillonite K10: An Efficient Organo- Heterogeneous Catalyst for Synthesis of Benzimidazole Derivatives
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DOI: 10.20944/preprints202007.0096.v1
Abstract: The use of alternative synthetic methods, in the face of traditional processes that do not conform to the principles of Green Chemistry, represent a problem in the pharmaceutical industry. The procedures for the synthesis of… read more here.
Keywords: montmorillonite k10; chemistry; synthesis benzimidazole; benzimidazole derivatives ... See more keywords