Synthesis of Benzoazepine Derivatives via Azide Rearrangement and Evaluation of Their Antianxiety Activities.
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DOI: 10.1021/acsmedchemlett.1c00275
Abstract: A new synthetic method for the construction of benzoazepine analogues has been developed employing ortho-arylmethylbenzyl azide derivatives as precursors using an azide rearrangement reaction. In this work, 14 benzoazepine compounds were successfully synthesized in moderate… read more here.
Keywords: antianxiety; synthesis benzoazepine; via azide; benzoazepine derivatives ... See more keywords