Structure–Activity Relationship of the Thiacalix[4]arenes Family with Sulfobetaine Fragments: Self-Assembly and Cytotoxic Effect against Cancer Cell Lines
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DOI: 10.3390/molecules27041364
Abstract: Regulating the structure of macrocyclic host molecules and supramolecular assemblies is crucial because the structure–activity relationship often plays a role in governing the properties of these systems. Herein, we propose and develop an approach to… read more here.
Keywords: sulfobetaine; cell; structure; activity ... See more keywords
Fluorescein-Labeled Thiacalix[4]arenes as Potential Theranostic Molecules: Synthesis, Self-Association, and Antitumor Activity
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DOI: 10.3390/pharmaceutics14112340
Abstract: In this paper, a series of thiacalix[4]arenes were synthesized as potential theranostic molecules for antitumor therapy. We propose an original strategy for the regioselective functionalization of thiacalix[4]arene with a fluorescent label to obtain antiangiogenic agent… read more here.
Keywords: potential theranostic; fluorescein labeled; thiacalix arenes; labeled thiacalix ... See more keywords