Articles with "triazole scaffolds" as a keyword



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Diversification of quinoline-triazole scaffolds with CORMs: Synthesis, in vitro and in silico biological evaluation against Plasmodium falciparum.

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Published in 2020 at "Journal of inorganic biochemistry"

DOI: 10.1016/j.jinorgbio.2020.111328

Abstract: A discrete series of tricarbonyl manganese and rhenium complexes conjugated to a quinoline-triazole hybrid scaffold were synthesised and their inhibitory activities evaluated against Plasmodium falciparum. In general, the complexes show moderate activity with improved inhibitory… read more here.

Keywords: quinoline triazole; diversification quinoline; plasmodium falciparum; plasmodium ... See more keywords